Synthesis of Tetrahydroquinoline derivatives via One Pot Multi-component (4+2) Cycloaddition (Povarov) Reaction

Pravin Chavan; Shivaji Jadhav; Megha Rai

doi:10.5958/0974-4150.2018.00024.X

Asian Journal of Research in Chemistry

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0974-4150 (Online)
0974-4169 (Print)

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Synthesis of Tetrahydroquinoline derivatives via One Pot Multi-component (4+2) Cycloaddition (Povarov) Reaction

Author(s): Pravin Chavan, Shivaji Jadhav, Megha Rai

Email(s): chemistryp141286@gmail.com

DOI: 10.5958/0974-4150.2018.00024.X

Address: Pravin Chavan1*, Shivaji Jadhav2, Megha Rai2
1Department of Chemistry, Doshi Vakil Arts and G.C.U.B. Science and Commerce College, Goregaon-Raigad, Maharashtra- India.
2Department of Chemistry, Dr. Rafiq Zakaria College for Women, Navkhanda, Jublee Park, Aurangabad Maharashtra- India.
*Corresponding Author

Published In: Volume - 11, Issue - 1, Year - 2018

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ABSTRACT:
In the presence of InCl3 as a catalyst one-pot (4p+2p) cycloaddition reaction of aromatic aldehydes, arylamines and DHF in ethanol proceeded smoothly to give tetrahydroquinoline derivatives (4a-4j) in excellent yields. Advantages of this method are shorter reaction time and biologically important.

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Cite this article:
Pravin Chavan, Shivaji Jadhav, Megha Rai. Synthesis of Tetrahydroquinoline derivatives via One Pot Multi-component (4+2) Cycloaddition (Povarov) Reaction. Asian J. Research Chem. 2018; 11(1):117-120. doi: 10.5958/0974-4150.2018.00024.X

Cite(Electronic):
Pravin Chavan, Shivaji Jadhav, Megha Rai. Synthesis of Tetrahydroquinoline derivatives via One Pot Multi-component (4+2) Cycloaddition (Povarov) Reaction. Asian J. Research Chem. 2018; 11(1):117-120. doi: 10.5958/0974-4150.2018.00024.X Available on: https://ajrconline.org/AbstractView.aspx?PID=2018-11-1-24

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Synthesis of Tetrahydroquinoline derivatives via One Pot Multi-component (4+2) Cycloaddition (Povarov) Reaction

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